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Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M4' and Ligand = 'BDBM81900'
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute Of Neurological Disorders And Stroke

Curated by PDSP Ki Database
LigandPNGBDBM81900(AQ-RA 741 | CAS_129989 | NSC_129989)
Affinity DataKi:  6.46nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute Of Neurological Disorders And Stroke

Curated by PDSP Ki Database
LigandPNGBDBM81900(AQ-RA 741 | CAS_129989 | NSC_129989)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-NMS from human muscarinic M4 receptor expressed in stable CHO-K1 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
National Institute Of Neurological Disorders And Stroke

Curated by PDSP Ki Database
LigandPNGBDBM81900(AQ-RA 741 | CAS_129989 | NSC_129989)
Affinity DataKi:  7.90nMAssay Description:Binding affinity to muscarinic M4 receptor (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
University Of Bologna

Curated by PDSP Ki Database
LigandPNGBDBM81900(AQ-RA 741 | CAS_129989 | NSC_129989)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed