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Found 1 Enz. Inhib. hit(s) with Target = 'Nuclear receptor ROR-alpha' and Ligand = 'BDBM50105919'
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50105919(CHEMBL3596632)
Affinity DataEC50:  8.36E+3nMAssay Description:Inverse agonist activity at Gal4 DNA binding domain-tagged human RORalpha expressed in HEK293T cells assessed as effect on receptor-mediated transcri...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed