Affinity DataEC50: 7.40E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx compound preincub...More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Antagonist activity at rat P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+4nMAssay Description:Antagonist activity at mouse P2X4 receptor by cell-based calcium influx assayMore data for this Ligand-Target Pair