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Found 1 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 7' and Ligand = 'BDBM50216377'
TargetP2X purinoceptor 7(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50216377(CHEMBL395737 | isoquinolinesulfon-5-yl-[3-oxo-3-(4...)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as effect on intracellular calcium influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed