Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform' and Ligand = 'BDBM50336405'
LigandPNGBDBM50336405(4-amino-2-methyl-N-(6-methylpyridin-3-yl)quinazoli...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of PI3Kalpha by fluorescene polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50336405(4-amino-2-methyl-N-(6-methylpyridin-3-yl)quinazoli...)
Affinity DataIC50:  112nMAssay Description:Inhibition of PI3Kalpha-phosphorylation at S473 residue in human BT20 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed