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Found 1 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50120727'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50120727(2-(2-Hydroxy-phenyl)-1,3,4,5-tetrahydro-azepino[5,...)
Affinity DataKi:  23nMAssay Description:In vitro inhibitory activity towards human poly(ADP-ribose) polymerase 1 (PARP-1).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed