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Found 4 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50300014'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50300014(2-(4-(Pyridin-4-yl)phenyl)-1H-benzimidazole-4-carb...)
Affinity DataKi:  2nMAssay Description:Inhibition of PARP1 using [3H]NAD+ by top count scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50300014(2-(4-(Pyridin-4-yl)phenyl)-1H-benzimidazole-4-carb...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of PARP1 by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50300014(2-(4-(Pyridin-4-yl)phenyl)-1H-benzimidazole-4-carb...)
Affinity DataEC50:  12nMAssay Description:Inhibition of PARP1 in human C41 cells by FITC-conjugated DAPI stainingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50300014(2-(4-(Pyridin-4-yl)phenyl)-1H-benzimidazole-4-carb...)
Affinity DataEC50:  12nMAssay Description:Inhibition of PARP1 in human C41 cells after 30 mins by cell-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed