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Found 1 Enz. Inhib. hit(s) with Target = 'Pro-glucagon' and Ligand = 'BDBM160577'
TargetPro-glucagon(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM160577(US9045389, 9)
Affinity DataKi:  38nM ΔG°:  -39.4kJ/molepH: 7.4 T: 2°CAssay Description:Full-length human GCGR (Accession Number: NM000160) subcloned into pcDNA3.1 was stably transfected into HEK293 cells (hGluc-1 HEK) and maintained und...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent