TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.01nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain (Wild type)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.01nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.01nMAssay Description:Binding of Indolactam-V(ILV) to wild-type Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC delta expressed in baculovirusMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 8.30nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C epsilon C1b domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 10.9nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (F13G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 10.9nMAssay Description:Binding of Indolactam-V(ILV) to mutant Protein kinase C delta C1b domain (Phe13 to Gly)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 25.3nMAssay Description:Binding of Indolactam-V(ILV) to mutant Protein kinase C delta C1b domain (Thr12 to Gly)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 25.3nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T12G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 66.2nMAssay Description:Binding of Indolactam-V(ILV) to mutant Protein kinase C delta C1b domain (Leu20 to Gly)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 66.2nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (L20G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 136nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C epsilon C1a domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 658nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T8G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 658nMAssay Description:Binding of Indolactam-V(ILV) to mutant Protein kinase C delta C1b domain (Tyr8 to Gly)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Binding of Indolactam-V(ILV) to mutant Protein kinase C delta C1b domain (Gln27 to Val)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (Q27V)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Binding affinity for Protein kinase C alpha C1a domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.90E+3nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C delta C1a domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 7.08E+3nMAssay Description:Binding of Indolactam-V(ILV) to mutant Protein kinase C delta C1b domain (Pro11 to Gly)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 7.08E+3nMAssay Description:Displacement of [3H]-PDBu from protein kinase C delta C1b domain mutant (P11G)More data for this Ligand-Target Pair