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Found 6 Enz. Inhib. hit(s) with Target = 'Putative P2Y purinoceptor 10' and Ligand = 'BDBM50096349'
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  28nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  28nMAssay Description:Agonist activity at P2Y10 (unknown origin) transfected in HEK293A cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  19nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  25nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse P2Y10 expressed in HEK293 cells co-transfected with AP-TGFalpha/Galphaq/i1 assessed as induction of ectodomain shedding of ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPutative P2Y purinoceptor 10(Mus musculus)
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50096349(CHEBI:52649 | CHEMBL1742484)
Affinity DataEC50:  25nMAssay Description:Agonist activity at mouse P2Y10 receptor expressed in HEK293A cells after 1.5 hrs by alkaline phosphatase tagged-TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed