Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha' and Ligand = 'BDBM50179115'
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179115((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataKi:  63nMAssay Description:Binding affinity to RXRalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50179115((2E,4E)-6-((6-tert-butyl-1,1-dimethyl-2,3-dihydro-...)
Affinity DataEC50:  123nMAssay Description:Transactivation of RXRalpha in CV1 cells by cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed