Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase 33' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase 33(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 36.3nMAssay Description:Inhibition of human STK33 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 33(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 38.4nMAssay Description:Inhibition of human STK33 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 33(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 1.80nMAssay Description:Binding constant for STK33 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 33(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataKd: 1.80nMAssay Description:Binding constant for full-length STK33More data for this Ligand-Target Pair