Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase Nek5' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase Nek5(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 76.3nMAssay Description:Inhibition of human NEK5 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek5(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 96.5nMAssay Description:Inhibition of human NEK5 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek5(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 810nMAssay Description:Binding constant for NEK5 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Nek5(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 810nMAssay Description:Binding constant for NEK5 kinase domainMore data for this Ligand-Target Pair