Found 7 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PAK 4' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Inner Mongolia Medical University
Curated by ChEMBL
Inner Mongolia Medical University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of protein kinase C epsilon expressed in Sf-9 cellsMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Inner Mongolia Medical University
Curated by ChEMBL
Inner Mongolia Medical University
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of recombinant human N-terminal GST-fused PAK4 (1 to 591 residues) expressed in baculovirus expression system using S2 as substrate measur...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Inner Mongolia Medical University
Curated by ChEMBL
Inner Mongolia Medical University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human PAK4 using RRRLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Inner Mongolia Medical University
Curated by ChEMBL
Inner Mongolia Medical University
Curated by ChEMBL
Affinity DataIC50: 27.9nMAssay Description:Inhibition of human PAK4 using RRRLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Inner Mongolia Medical University
Curated by ChEMBL
Inner Mongolia Medical University
Curated by ChEMBL
Affinity DataKd: 6.30nMAssay Description:Binding constant for PAK4 kinase domainMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Inner Mongolia Medical University
Curated by ChEMBL
Inner Mongolia Medical University
Curated by ChEMBL
Affinity DataKd: 8nMAssay Description:Average Binding Constant for PAK4; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase PAK 4(Homo sapiens (Human))
Inner Mongolia Medical University
Curated by ChEMBL
Inner Mongolia Medical University
Curated by ChEMBL
Affinity DataKd: 6.30nMAssay Description:Binding constant for PAK4 kinase domainMore data for this Ligand-Target Pair