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Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PLK1' and Ligand = 'BDBM50402026'
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50402026(CHEMBL2205457)
Affinity DataKi:  14nMAssay Description:Inhibition of recombinant GST-tagged PLK1 using biotin-ahx-AKMETTFYDDALNASFLPSEKKK-amide as substrate after 30 mins by scintillation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50402026(CHEMBL2205457)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of PLK1 in human MIAPaCa2 cells after 48 hrs by MTT assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed