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Found 4 Enz. Inhib. hit(s) with Target = 'Serine-protein kinase ATM' and Ligand = 'BDBM50098126'
TargetSerine-protein kinase ATM(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50098126(2-(morpholin-4-yl)-benzo[h]chromen-4-one | 2-Morph...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ATMChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine-protein kinase ATM(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50098126(2-(morpholin-4-yl)-benzo[h]chromen-4-one | 2-Morph...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of full length recombinant ATM after 24 hrs by radiometric phosphate incorporation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine-protein kinase ATM(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50098126(2-(morpholin-4-yl)-benzo[h]chromen-4-one | 2-Morph...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ATM kinase using rabbit polyclonal antiseraMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine-protein kinase ATM(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50098126(2-(morpholin-4-yl)-benzo[h]chromen-4-one | 2-Morph...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of Mutated in ataxia telangiectasia protein ATM kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed