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Found 2 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50040283'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50040283(3-Chloro-6-dimethylamino-6-methyl-8-phenyl-5,6,7,8...)
Affinity DataIC50:  0.290nMAssay Description:Binding affinity against sigma receptor from guinea pig brain (minus cerebellum) homogenates, using the novel [3H]-(+/-)-4 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University Of North Carolina

Curated by ChEMBL
LigandPNGBDBM50040283(3-Chloro-6-dimethylamino-6-methyl-8-phenyl-5,6,7,8...)
Affinity DataIC50:  3.40E+3nMAssay Description:Binding affinity against sigma receptor from guinea pig brain (minus cerebellum) homogenates, using [3H]ditolylguanidine (DTG) as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed