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Found 5 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50374606'
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by PDSP Ki Database
LigandPNGBDBM50374606(CHEMBL405925 | US9604926, Compound CM-124 | US9724...)
Affinity DataKi:  5.22nMAssay Description:Displacement of [3H](+)-pentazocine from opioid sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by PDSP Ki Database
LigandPNGBDBM50374606(CHEMBL405925 | US9604926, Compound CM-124 | US9724...)
Affinity DataKi:  5.22nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
The University Of Mississippi

US Patent
LigandPNGBDBM50374606(CHEMBL405925 | US9604926, Compound CM-124 | US9724...)
Affinity DataKi:  5.22nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(Mus musculus (Mouse))
The University Of Mississippi

US Patent
LigandPNGBDBM50374606(CHEMBL405925 | US9604926, Compound CM-124 | US9724...)
Affinity DataKi:  5.22nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSigma non-opioid intracellular receptor 1(RAT)
The University Of Mississippi

Curated by PDSP Ki Database
LigandPNGBDBM50374606(CHEMBL405925 | US9604926, Compound CM-124 | US9724...)
Affinity DataKi:  5.22nMAssay Description:Compounds were evaluated for σ-1 and σ-2 binding in rat brain homogenates. Twelve concentrations of each test ligand (0.001-1,000 nM) were ...More data for this Ligand-Target Pair
In DepthDetails US Patent