Found 36 Enz. Inhib. hit(s) with Target = 'Sodium-dependent noradrenaline transporter' and Ligand = 'BDBM50084717'
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 182nMAssay Description:Inhibition of [3H]DA uptake in human NET expressed in COS1 cell membraneMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 190nMAssay Description:Inhibition of reuptake of [3H]-NE (20 nM) by norepinephrine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 264nMAssay Description:Compound was evaluated for inhibition of [3H]NE uptake in HEK-hNET cells expressing Human norepinephrine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 500nMAssay Description:Displacement of [125I]RTI-55 from human NET expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 830nMAssay Description:Displacement of [125I]RTI55 from cloned human NET expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 887nMAssay Description:Displacement of [125I]RTI55 from human NET expressed in COS1 cell membraneMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.12E+3nMAssay Description:Displacement of [125I]RTI55 from human recombinant NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.12E+3nMAssay Description:Displacement of [125I]RTI55 from human NET expressed in HEK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.74E+3nMAssay Description:Compound was evaluated for binding affinity using [125I]RTI-55 as a radioligand in HEK-hNET cells expressing human norepinephrine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.77E+3nMAssay Description:Binding affinity at the norepinephrine transporter was measured using [125I]RTI-55 as a radioligandMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.77E+3nMAssay Description:Inhibition of [125I]RTI-55 binding to norepinephrine transporter (NET) expressed in HEK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.94E+3nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.99E+3nMAssay Description:Displacement of [3H]nisoxetine from norepinephrine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.99E+3nMAssay Description:Displacement of [3H]nisoxetine from NETMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.99E+3nMAssay Description:Displacement of [3H]nisoxetine from NETMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.99E+3nMAssay Description:Displacement of [3H]nisoxetine from human NETMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 1.99E+3nMAssay Description:Displacement of [3H]nisoxetine from NETMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 2.15E+3nMAssay Description:Displacement of [125I]RTI-55 from human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 2.38E+3nMAssay Description:Displacement of [125I]RTI-55 from human recombinant NET expressed in HEK293 cells by scintillation countingMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataKi: 2.70E+3nMAssay Description:Binding affinity against norepinephrine cloned human transporter using 40-80 pM [125I]RTIMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Inhibition of [3H]NE uptake into human NET expressing HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of [3H]- NE uptake in HEK cells expressing norepinephrine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of [3H]NE reuptake by human norepinephrine transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 232nMAssay Description:Inhibition of [3H]NE reuptake at human NET expressed in HEK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 233nMAssay Description:Inhibition of NE uptake in HEK cells expressing human noradrenaline transporter (hNET)More data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 378nMAssay Description:Inhibition of [3H] norepinephrine uptake into human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 385nMAssay Description:Inhibition of [3H]norepinephrine reuptake at human NET expressed in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 462nMAssay Description:Inhibition of [3H]norepinephrine uptake in HEK293 cells expressing human norepinephrine transporterMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 835nMAssay Description:Inhibition of [3H]NE from human recombinant NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of rat NET-mediated norepinephrine uptake in CHO cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of [3H]norepinephrine reuptake at human NET expressed in HEK cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of [3H]norepinephrine uptake at human NET expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 2.99E+3nMAssay Description:Displacement of [125I]RTI-55 from human Norepinephrine transporter expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Displacement of [3H]nisoxetine from NETMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Displacement of [3H]nisoxetine from NETMore data for this Ligand-Target Pair
TargetSodium-dependent noradrenaline transporter(Homo sapiens (Human))
University Of Aarhus
Curated by ChEMBL
University Of Aarhus
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Displacement of [3H]nisoxetine from human NETMore data for this Ligand-Target Pair