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Found 11 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 3' and Ligand = 'BDBM50065453'
TargetSomatostatin receptor type 3(MOUSE)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  107nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  107nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(MOUSE)
Sandoz Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  108nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  126nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  126nMAssay Description:Binding affinity towards human Somatostatin receptor type 3 (sst3) using Tyr11-[125I]-SRIF as radioligand was determined in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  129nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst3) expressed in CHO-K1 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  148nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  148nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  457nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKi:  457nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Novartis Pharma

Curated by PDSP Ki Database
LigandPNGBDBM50065453((5S,8S,11S,14R,17S,19aS)-11-(4-Amino-butyl)-5,17-d...)
Affinity DataKd:  525nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst3) expressed in CHO cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed