Affinity DataKi: 0.380nMAssay Description:Inhibitory constant against human sst5 receptor at a dose of 10 uMMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair