Found 26 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50000041' 
Affinity DataKi: 0.170nMAssay Description:In vitro inhibitory activity against human NK1 receptor was determinedMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 0.170nMAssay Description:Evaluated for the binding affinity towards NK1 receptor in the striatal membranes of guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Evaluated for the binding affinity towards NK1 receptor in the striatal membranes of guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:Binding affinity to Tachykinin receptor 1 stably expressed in chinese hamster ovary (CHO) cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.251nMAssay Description:In vitro binding affinity against human NK1 receptor expressed in CHO cells using [3H]-substance P as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:Binding affinity was carried out with NK 1 receptors from U-373MG human astrocytoma cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 0.398nMAssay Description:Compound was evaluated for binding affinity towards neurokinin NK1 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:In vitro binding affinity for the Tachykinin receptor 1 in human IM-9 cell using [125I]-BH-SP of the compound.More data for this Ligand-Target Pair
Affinity DataKi: 0.480nMAssay Description:In vitro binding affinity for the Tachykinin receptor 1 in human IM-9 cell using [125I]-BH-SP of the compound.More data for this Ligand-Target Pair
Affinity DataKi: 0.794nMAssay Description:Binding affinity measured by displacement of tritiated radiolabeled substance P from cloned human NK1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro binding affinity of the compound towards human NK-1 receptor in IM-9 cells using [3H]-SP of substance P antagonistMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:In vitro binding affinity for the Tachykinin receptor 1 in human IM-9 cell using [125I]BH-SP of the compound.More data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Antagonist activity at NK1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Binding affinity was measured against the Tachykinin receptor 1 in human IM-9 cells using [3H]SP as ligand.More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of [125I]-BH-Substance P binding to tachykinin receptor 1 in human IM-9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.490nMAssay Description:Antagonist activity for Tachykinin receptor 1 as displacement of [3H]-Substance P in human IM-9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in CHO cells was measured by its ability to displace [125I]- Tyr-8 substance P.More data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Binding affinity towards Neurokinin -1(NK-1) receptor of human by using [125I]- Tyr8 substance P as a radioligand in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Displacement of [125 I]-Tyr8 SP from the cloned human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Displacement of [125I]-labeled SP from human Tachykinin receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Inhibition of substance P binding to Tachykinin receptor 1 in Chinese hamster ovary cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I]- Substance P from human Neurokinin 1 (hNK1) receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.630nMAssay Description:Displacement of [3H]substance P from NK1 human receptor expressed in IM9 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Binding affinity of the compound towards human Tachykinin receptor 1 by the displacement of [125I]- Substance P in CHO CellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.90nMAssay Description:In vitro binding affinity against Tachykinin receptor 1 in guinea pig ileum using organ bath assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.320nMAssay Description:Evaluated for the binding affinity towards NK1 receptor in the striatal membranes of guinea pigMore data for this Ligand-Target Pair
