Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Substance-P receptor' and Ligand = 'BDBM50281980'
TargetSubstance-P receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50281980((2S,3S)-2-Benzhydryl-3-(3-methyl-benzyloxy)-1-aza-...)
Affinity DataIC50:  20.9nMAssay Description:Binding affinity was measured against the Tachykinin receptor 1 in CHO-expressed hNK1 using [125I]SP.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50281980((2S,3S)-2-Benzhydryl-3-(3-methyl-benzyloxy)-1-aza-...)
Affinity DataIC50:  21nMAssay Description:Displacement of [125]Substance P Binding from human Neurokinin NK1 receptor in CHO CellsMore data for this Ligand-Target Pair
In DepthDetails Article