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Found 2 Enz. Inhib. hit(s) with Target = 'Thymidine kinase, cytosolic' and Ligand = 'BDBM50118489'
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50118489(1-(4-Hydroxy-5-trityloxymethyl-tetrahydro-furan-2-...)
Affinity DataIC50:  7.80E+3nMAssay Description:Compound was evaluated for inhibitory effect against phosphorylation of [methyl-3H]dThd by HSV-1 Thymidine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine kinase, cytosolic(Homo sapiens (Human))
Instituto De Qu£Mica M£Dica (Csic)

Curated by ChEMBL
LigandPNGBDBM50118489(1-(4-Hydroxy-5-trityloxymethyl-tetrahydro-furan-2-...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibitory effect against phosphorylation of [methyl-3H]dThd by Thymidine Kinase 2 (TK-2)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed