Found 3 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1' and Ligand = 'BDBM61009'
TargetTransient receptor potential cation channel subfamily A member 1(Mus musculus)
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataEC50: 1.30E+5nMAssay Description:Agonist activity at TRPA1 channel in mouse dorsal root ganglion cells assessed as increase in intracellular calcium influx by radiometric Ca2+ imagin...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Mus musculus)
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataEC50: 2.58E+3nMAssay Description:Agonist activity at mouse TRPA1 channel expressed in HEK293 cells assessed as increase in intracellular calcium influxMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataEC50: 590nMAssay Description:Agonist activity at human TRPA1 channel expressed in HEK293 cells assessed as increase in intracellular calcium influxMore data for this Ligand-Target Pair