Found 15 Enz. Inhib. hit(s) with Target = 'Translocator protein' and Ligand = 'BDBM50122293' TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.0430nMAssay Description:In vitro binding affinity for PBR (peripheral benzodiazepine receptor) in rat brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.0726nMAssay Description:Displacement of [3H]PK11195 from rat PBR receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.0726nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Displacement of [11C]DAA1106 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.188nMAssay Description:In vitro binding affinity for PBR (peripheral benzodiazepine receptor) in monkey brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Inhibition of human TSPOMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.242nMAssay Description:Displacement of [3H]PK11195 from human PBR receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.242nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataKi: 0.430nMAssay Description:Displacement of [3H]PK11195 from TSPO in Wistar rat heart incubated for 15 minsMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataIC50: 0.280nMAssay Description:Inhibition of TSPO receptor (unknown origin)More data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Displacement of [11C]PK-11195 from PBR in Sprague-Dawley rat brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Displacement of [11C]DAA1106 from PBR in Sprague-Dawley rat brainMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences
Curated by ChEMBL
National Institute Of Radiological Sciences
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:In vitro displacement of [11C]-DAA1106 from PBR (peripheral benzodiazepine receptor) of rat brainMore data for this Ligand-Target Pair
