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Found 2 Enz. Inhib. hit(s) with Target = 'Transmembrane domain-containing protein TMIGD3' and Ligand = 'BDBM50163878'
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50163878(CHEMBL3799738)
Affinity DataKi:  60nMAssay Description:Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyl-uronamide from human adenosine A3 receptor expressed in CHO cell membranes incub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransmembrane domain-containing protein TMIGD3(Homo sapiens (Human))
National Institute Of Diabetes And Digestive And Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50163878(CHEMBL3799738)
Affinity DataEC50:  27nMAssay Description:Agonist activity at recombinant human adenosine A3 receptor expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP accumulation p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed