Found 7 Enz. Inhib. hit(s) with Target = 'Vesicular acetylcholine transporter' and Ligand = 'BDBM50018078' 
Affinity DataKi: 9.90nMAssay Description:The binding affinity of a compound to VAChT was measured by competition against the binding of 5 nM [3H]Vesamicol to postnuclear supernatant prepared...More data for this Ligand-Target Pair
Affinity DataKi: 32.9nMAssay Description:Displacement of [125I]O-iodo-trans-decalinvesamicol from VAChT in Sprague-Dawley rat cerebral membrane after 1 hr by gamma countingMore data for this Ligand-Target Pair
Affinity DataKi: 33.9nMAssay Description:Displacement of (-)-[3H]vesamicol from VAChT in Sprague-Dawley rat cerebral membrane after 60 mins by liquid scintillation counting in presence of DT...More data for this Ligand-Target Pair
Affinity DataKi: 49nMAssay Description:Displacement of (-)-[3H]vesamicol from rat VAChT expressed in rat PC12 cell membranes after 60 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetVesicular acetylcholine transporter(Torpedo californica)
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Displacement of [3H]-Vesamicol from Vesamicol receptor of Torpedo californicaMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of active transport of [3H]acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of active transport of [3H]-Acetylcholine using purified Torpedo californica synaptic vesiclesMore data for this Ligand-Target Pair
