Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with Target = 'Plasmin' and Monomerid = 14155
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Celera

Curated by ChEMBL
LigandPNGBDBM14155(APC-7136 | CHEMBL64708 | N-(4-CARBAMIMIDOYL-PHENYL...)
Affinity DataKi:  2.70E+3nMAssay Description:Inhibition of urokinase-type plasminogen activator (microPa)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Celera

Curated by ChEMBL
LigandPNGBDBM14155(APC-7136 | CHEMBL64708 | N-(4-CARBAMIMIDOYL-PHENYL...)
Affinity DataKi:  3.80E+3nM ΔG°:  -30.6kJ/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Axys Pharmaceutical

LigandPNGBDBM14155(APC-7136 | CHEMBL64708 | N-(4-CARBAMIMIDOYL-PHENYL...)
Affinity DataKi:  6.60E+3nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Celera

Curated by ChEMBL
LigandPNGBDBM14155(APC-7136 | CHEMBL64708 | N-(4-CARBAMIMIDOYL-PHENYL...)
Affinity DataKi:  1.00E+4nMAssay Description:Activation of tissue plasminogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Celera

Curated by ChEMBL
LigandPNGBDBM14155(APC-7136 | CHEMBL64708 | N-(4-CARBAMIMIDOYL-PHENYL...)
Affinity DataKi:  1.20E+4nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Axys Pharmaceutical

LigandPNGBDBM14155(APC-7136 | CHEMBL64708 | N-(4-CARBAMIMIDOYL-PHENYL...)
Affinity DataKi:  9.00E+4nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed