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Found 3 Enz. Inhib. hit(s) with Target = 'Plasmin' and Monomerid = 16140
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Pfizer

LigandPNGBDBM16140(1-guanidino-7-sulfonamidoisoquinoline 14 | 3-({4-c...)
Affinity DataKi:  58nM ΔG°:  -43.0kJ/molepH: 8.1 T: 2°CAssay Description:Ki values for compounds were calculated by incubation of each enzyme with its substrate and various compound concentrations. Absorbance was read at 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Pfizer

LigandPNGBDBM16140(1-guanidino-7-sulfonamidoisoquinoline 14 | 3-({4-c...)
Affinity DataKi: >1.00E+5nMAssay Description:Ki values for compounds were calculated by incubation of each enzyme with its substrate and various compound concentrations. Absorbance was read at 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Pfizer

LigandPNGBDBM16140(1-guanidino-7-sulfonamidoisoquinoline 14 | 3-({4-c...)
Affinity DataKi: >1.00E+5nMAssay Description:Ki values for compounds were calculated by incubation of each enzyme with its substrate and various compound concentrations. Absorbance was read at 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed