Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Plasmin' and Monomerid = 16153
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Pfizer

LigandPNGBDBM16153(1-({4-chloro-1-[(diaminomethylidene)amino]isoquino...)
Affinity DataKi:  7.40nMAssay Description:Ki values for compounds were calculated by incubation of each enzyme with its substrate and various compound concentrations. Absorbance was read at 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Pfizer

LigandPNGBDBM16153(1-({4-chloro-1-[(diaminomethylidene)amino]isoquino...)
Affinity DataKi:  1.60E+4nMAssay Description:Ki values for compounds were calculated by incubation of each enzyme with its substrate and various compound concentrations. Absorbance was read at 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Pfizer

LigandPNGBDBM16153(1-({4-chloro-1-[(diaminomethylidene)amino]isoquino...)
Affinity DataKi: >1.00E+5nMAssay Description:Ki values for compounds were calculated by incubation of each enzyme with its substrate and various compound concentrations. Absorbance was read at 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed