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Found 4 Enz. Inhib. hit(s) with Target = 'Plasmin' and Monomerid = 16175
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM16175(CHEMBL108468 | UKI-1 | ethyl 4-(3-carbamimidoyl-N-...)
Affinity DataKi:  410nM ΔG°:  -36.5kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM16175(CHEMBL108468 | UKI-1 | ethyl 4-(3-carbamimidoyl-N-...)
Affinity DataKi:  960nMAssay Description:Tested for inhibition of plasminogen activator urokinase (microPa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM16175(CHEMBL108468 | UKI-1 | ethyl 4-(3-carbamimidoyl-N-...)
Affinity DataKi:  1.20E+3nMAssay Description:Tested for inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Max-Planck-Institut Fuer Biochemie

LigandPNGBDBM16175(CHEMBL108468 | UKI-1 | ethyl 4-(3-carbamimidoyl-N-...)
Affinity DataKi:  4.90E+3nM ΔG°:  -30.3kJ/molepH: 8.0 T: 2°CAssay Description:The measurements were carried out on a microplate reader. Two concentrations of the substrate and five concentrations of the inhibitor were used in t...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed