Affinity DataKi: 19.3nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A2B receptor expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]ZM-241385 from human A2B receptor expressed in HEK-293 cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Selectivity for recombinant human adenosine A2b receptorMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Antagonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of NECA-stimulated [3H]cAMP production by scintilla...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of human recombinant adenosine receptor A2bMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of human adenosine 2B receptorMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]DPCPX from human Adenosine A2B receptor expressed in HEK293 cells after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]DPCPX from human A2BAR expressed in HEK293 cell membrane incubated for 30 mins by microbeta trilux scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cell membranes incubated for 60 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]DPCPX from human recombinant A2B receptor expressed in human HEK293 cell membranes incubated for 30 mins by radioligand binding c...More data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]DPCPX from human recombinant A2B receptor expressed in human HEK293 cell membranes incubated for 30 mins by radioligand binding c...More data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inverse agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of cAMP accumulation measured after 150 mins i...More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inverse agonist activity at human adenosine A2B receptor expressed in CHO cells assessed as inhibition of cAMP accumulation measured after 150 mins i...More data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Displacement of PSB-12105 from recombinant human adenosine A2B receptor expressed in CHO cell membranes preincubated for 30 mins followed by PSB-1210...More data for this Ligand-Target Pair