Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Peptide Deformylase' and Monomerid = 21685
TargetPeptide deformylase(Haemophilus influenzae)
Gsk

LigandPNGBDBM21685(N-hydroxy-N-[3-(6-methylpyridin-2-yl)propyl]formam...)
Affinity DataIC50:  1.04E+3nMpH: 7.6 T: 2°CAssay Description:Enzyme assay was carried out in 96-well microtiter plates with a SpectraMax plate reader (Molecular Devices Corp.). PDF activity was measured using a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Gsk

LigandPNGBDBM21685(N-hydroxy-N-[3-(6-methylpyridin-2-yl)propyl]formam...)
Affinity DataIC50:  1.09E+3nMpH: 7.6 T: 2°CAssay Description:Enzyme assay was carried out in 96-well microtiter plates with a SpectraMax plate reader (Molecular Devices Corp.). PDF activity was measured using a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Streptococcus pneumoniae (strain ATCC BAA-255 / R6...)
Gsk

LigandPNGBDBM21685(N-hydroxy-N-[3-(6-methylpyridin-2-yl)propyl]formam...)
Affinity DataIC50:  2.20E+3nMpH: 7.6 T: 2°CAssay Description:Enzyme assay was carried out in 96-well microtiter plates with a SpectraMax plate reader (Molecular Devices Corp.). PDF activity was measured using a...More data for this Ligand-Target Pair
TargetPeptide deformylase(Escherichia coli (strain K12))
Gsk

LigandPNGBDBM21685(N-hydroxy-N-[3-(6-methylpyridin-2-yl)propyl]formam...)
Affinity DataIC50:  2.80E+3nMpH: 7.6 T: 2°CAssay Description:Enzyme assay was carried out in 96-well microtiter plates with a SpectraMax plate reader (Molecular Devices Corp.). PDF activity was measured using a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed