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Found 1 Enz. Inhib. hit(s) with Target = 'Adenosine Receptor A1' and Monomerid = 25399
TargetAdenosine receptor A1(Homo sapiens (Human))
Monash University

LigandPNGBDBM25399(Bivalent derivative, 18 | N-[5-(1-{9-[(2R,3R,4S,5R...)
Affinity DataKi:  1.91E+3nM ΔG°:  -32.3kJ/molepH: 7.4 T: 2°CAssay Description:The displacement of [3H]DPCPX binding from the A1AR was determined using DDT1 MF-2 cell membranes. Nonspecific binding was determined in parallel ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed