TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 7.60nMAssay Description:Inhibition of human IRR using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.80nMAssay Description:Inhibition of human IR using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of human IRR using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of IR (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 17.7nMAssay Description:Inhibition of human IR using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Inhibition of INSR (unknown origin) incubated for 1 hr by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetInsulin receptor(Mus musculus)
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of Insulin receptor kinase in P19 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: <300nMAssay Description:Inhibition of Insulin receptorMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 81nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair
TargetInsulin receptor-related protein(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 81nMAssay Description:Binding constant for INSRR kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 73nMAssay Description:Average Binding Constant for INSR; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding constant for INSR kinase domainMore data for this Ligand-Target Pair