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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Src' and Monomerid = 4097   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Proto-oncogene tyrosine-protein kinase Src


(Homo sapiens (Human))
BDBM4097
PNG
(9-benzoyl-9H-carbazole-1,2,6,7-tetrol | Carbazole ...)
Show SMILES Oc1cc2n(C(=O)c3ccccc3)c3c(O)c(O)ccc3c2cc1O
Show InChI InChI=1S/C19H13NO5/c21-14-7-6-11-12-8-15(22)16(23)9-13(12)20(17(11)18(14)24)19(25)10-4-2-1-3-5-10/h1-9,21-24H
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
PC cid
PC sid
UniChem

Patents


Similars

Article
PubMed
n/an/a 900n/an/an/an/an/an/a



Pfizer



Assay Description
IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...


J Med Chem 37: 2224-31 (1994)


Article DOI: 10.1021/jm00040a015
BindingDB Entry DOI: 10.7270/Q27M0648
More data for this
Ligand-Target Pair