Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Thromboxane A2 receptor' and Monomerid = 50002759
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002759(5-(2-Benzenesulfonylamino-ethylsulfanyl)-5,11-dihy...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002759(5-(2-Benzenesulfonylamino-ethylsulfanyl)-5,11-dihy...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity at TXA2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed