Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Thromboxane A2 receptor' and Monomerid = 50002776
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002776(11-[2-(2-Nitro-benzenesulfonylamino)-ethylsulfanyl...)
Affinity DataKi:  15nMAssay Description:Inhibition of Shh signaling in mouse Shh-light2 cells by Gli-dependent firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50002776(11-[2-(2-Nitro-benzenesulfonylamino)-ethylsulfanyl...)
Affinity DataKi:  15nMAssay Description:Binding affinity at TXA2 receptor by measuring its ability to displace [3H]-U-46,619 from guinea pig plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed