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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Phosphodiesterase 2A' and Monomerid = 50007217   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Homo sapiens phosphodiesterase 2A (PDE2A)


(Homo sapiens (Human))
BDBM50007217
PNG
(7-Chloro-1,3,9,9a-tetrahydro-imidazo[4,5-b]quinoli...)
Show SMILES Clc1ccc2Nc3[nH]c(=O)[nH]c3Cc2c1
Show InChI InChI=1S/C10H8ClN3O/c11-6-1-2-7-5(3-6)4-8-9(12-7)14-10(15)13-8/h1-3,12H,4H2,(H2,13,14,15)
PDB

UniProtKB/SwissProt

antibodypedia
GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 8.00E+4n/an/an/an/an/an/a



Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Inhibition of cGMP hydrolysis by human platelet phosphodiesterase


J Med Chem 34: 2906-16 (1991)


Article DOI: 10.1021/jm00113a033
BindingDB Entry DOI: 10.7270/Q20P0Z03
More data for this
Ligand-Target Pair