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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine Receptor A2A' and Monomerid = 50037422
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50037422(CHEMBL17123 | [4-(1,3-Dibutyl-2,6-dioxo-2,3,6,7-te...)
Affinity DataKi:  874nMAssay Description:Displacement of [3H]-CGS- 21680 from adenosine A2a receptors of rat striatal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50037422(CHEMBL17123 | [4-(1,3-Dibutyl-2,6-dioxo-2,3,6,7-te...)
Affinity DataKi:  874nMAssay Description:Antagonist activity against adenosine A2A receptor in rat striatal membrane in presence of [3H]-CGS-21,680 radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
National Institute Of Diabetes

Curated by ChEMBL
LigandPNGBDBM50037422(CHEMBL17123 | [4-(1,3-Dibutyl-2,6-dioxo-2,3,6,7-te...)
Affinity DataKi:  2.54E+3nMAssay Description:Antagonist activity against recombinant human adenosine A2A receptor expressed in HEK-293 cells in presence of [125I]-iodo-ZM241385 radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed