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Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL' and Monomerid = 50045528
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50045528(CHEMBL57553 | N-(4-Pyridin-3-yl-pyrimidin-2-yl)-be...)
Affinity DataIC50:  700nMAssay Description:Inhibition of v-Abl tyrosine kinase.More data for this Ligand-Target Pair
In DepthDetails Article
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
The First People'S Hospital Of Hangzhou

Curated by ChEMBL
LigandPNGBDBM50045528(CHEMBL57553 | N-(4-Pyridin-3-yl-pyrimidin-2-yl)-be...)
Affinity DataIC50:  708nMAssay Description:Inhibition of BCR-ABL kinase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1/ABL2(Homo sapiens (Human))
Mcgill University/Royal Victoria Hospital

Curated by ChEMBL
LigandPNGBDBM50045528(CHEMBL57553 | N-(4-Pyridin-3-yl-pyrimidin-2-yl)-be...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Abl tyrosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed