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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50048167   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Progesterone receptor


(Homo sapiens (Human))
BDBM50048167
PNG
((3,4-Dichloro-phenyl)-(3-phenyl-5,6-dihydro-4H-pyr...)
Show SMILES Clc1ccc(cc1Cl)C(=S)N1CCCC(=N1)c1ccccc1
Show InChI InChI=1S/C17H14Cl2N2S/c18-14-9-8-13(11-15(14)19)17(22)21-10-4-7-16(20-21)12-5-2-1-3-6-12/h1-3,5-6,8-9,11H,4,7,10H2
PDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Patents


Similars

Article
PubMed
n/an/a 18n/an/an/an/an/an/a



R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL


Assay Description
Binding affinity against Progesterone receptor in human TE85 osteosarcoma cells was determined using (Z)-[125I]-17-alpha-(2-iodovinyl)-19-nor-testost...


J Med Chem 38: 4880-4 (1996)


Article DOI: 10.1021/jm00025a004
BindingDB Entry DOI: 10.7270/Q2KP82SZ
More data for this
Ligand-Target Pair