Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50049507
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049507(5-Bromo-2-((1S,2R,4R)-2,4-dimethyl-6-methylene-cyc...)
Affinity DataKi:  84nMAssay Description:Binding affinity determined for human Progesterone receptor A isoformMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049507(5-Bromo-2-((1S,2R,4R)-2,4-dimethyl-6-methylene-cyc...)
Affinity DataIC50:  350nMAssay Description:Antagonistic potency to the human progesterone receptor measured in the T-47D alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049507(5-Bromo-2-((1S,2R,4R)-2,4-dimethyl-6-methylene-cyc...)
Affinity DataIC50:  985nMAssay Description:Concentration required to give half-maximal inhibition against human Progesterone receptor B isoform in co-transfected CV-1 cell lines.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed