Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50049513
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049513(5-Bromo-4-methoxy-2-((1R,2S)-2-methyl-6-methylene-...)
Affinity DataKi:  71nMAssay Description:Binding affinity determined for human Progesterone receptor A isoformMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049513(5-Bromo-4-methoxy-2-((1R,2S)-2-methyl-6-methylene-...)
Affinity DataIC50:  300nMAssay Description:Antagonistic potency to the human progesterone receptor measured in the T-47D alkaline phosphatase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50049513(5-Bromo-4-methoxy-2-((1R,2S)-2-methyl-6-methylene-...)
Affinity DataIC50:  1.05E+3nMAssay Description:Concentration required to give half-maximal inhibition against human Progesterone receptor B isoform in co-transfected CV-1 cell lines.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed