Found 5 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 4' and Monomerid = 50060137
Affinity DataEC50: 7.20E+3nMAssay Description:Agonist activity against Metabotropic glutamate receptor 4 expressed in HEK 293 cells was evaluated by measuring total inositol phosphate accumulatio...More data for this Ligand-Target Pair
Affinity DataEC50: 7.00E+3nMAssay Description:Agonistic activity at Metabotropic glutamate receptor 4 expressed in mammalian cells by GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+3nMAssay Description:Agonist activity at mGlu4 (unknown origin) expressed in HEK293 cells coexpressing chimeric Gq/i protein assessed as [3H]inositol phosphate accumulati...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Universite Paris Descartes
Curated by ChEMBL
Universite Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 1.74E+3nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells co-transfected with G-protein alpha and EAAC1 assessed as increase in intracellular ...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Universite Paris Descartes
Curated by ChEMBL
Universite Paris Descartes
Curated by ChEMBL
Affinity DataEC50: 7.20E+3nMAssay Description:Activity at rat mGluR4 receptor measured as intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair