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Found 3 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50062403
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062403(5-(4-Fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H...)
Affinity DataKi:  5.30nMAssay Description:The binding affinity of the compound was determined on Human progesterone receptor (hPR-A) using progesterone as radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062403(5-(4-Fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H...)
Affinity DataIC50:  342nMAssay Description:Antagonistic activity was determined in Human progesterone receptor(hPR) of CV-1 cells in cotransfection assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50062403(5-(4-Fluoro-phenyl)-2,2,4-trimethyl-2,5-dihydro-1H...)
Affinity DataEC50:  8nMAssay Description:Agonistic activity to the human progesterone receptor(hPR)assayed in CV-1 cells in cotransfection assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed