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Found 3 Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Monomerid = 50071885
TargetGlucagon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50071885(4-[2-(4-Chloro-phenyl)-5-(4-fluoro-phenyl)-3H-imid...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human glucagon receptor expressed in CHO cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlucagon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50071885(4-[2-(4-Chloro-phenyl)-5-(4-fluoro-phenyl)-3H-imid...)
Affinity DataIC50:  400nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50071885(4-[2-(4-Chloro-phenyl)-5-(4-fluoro-phenyl)-3H-imid...)
Affinity DataIC50:  3.20E+3nMAssay Description:Affinity for human glucagon receptor in presence of Mg2+More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed