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Found 3 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50072021
TargetProgesterone receptor(Homo sapiens (Human))
Scientific Computing

Curated by ChEMBL
LigandPNGBDBM50072021(2,2,4-Trimethyl-2,10-dihydro-1H-pyrido[2,3-b]carba...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]progesterone from Progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Scientific Computing

Curated by ChEMBL
LigandPNGBDBM50072021(2,2,4-Trimethyl-2,10-dihydro-1H-pyrido[2,3-b]carba...)
Affinity DataKi:  113nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Scientific Computing

Curated by ChEMBL
LigandPNGBDBM50072021(2,2,4-Trimethyl-2,10-dihydro-1H-pyrido[2,3-b]carba...)
Affinity DataIC50:  59nMAssay Description:Binding affinity against human progesterone receptor-A (hPR-A)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed