Found 3 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Monomerid = 50072228
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Melbourne
Curated by PDSP Ki Database
University Of Melbourne
Curated by PDSP Ki Database
Affinity DataIC50: 4.70nMAssay Description:Binding affinity against muscarinic receptor in rat brain membranes using oxotremorine-M as ligandMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Melbourne
Curated by PDSP Ki Database
University Of Melbourne
Curated by PDSP Ki Database
Affinity DataEC50: 16nMAssay Description:Stimulation of phosphoinositide hydrolysis in A9L cells expressing human m1 receptorMore data for this Ligand-Target Pair